Table 1

Cardioselectivity of β-blockers

Cardioselective β-blockersRelative β1/β2 selectivityUsual dose range (mg/day) (frequency per day)
Celiprolol69200–400 (1)
Metoprolol7450–200 (1–2)
Betaxolol9310–20 (1)
Bisoprolol1032.5–10 (1)
Nebivolol3215–40 (1)